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Title A development of chimeric VEGFR2 TK inhibitor based on two ligand conformers from PDB: 1Y6A complex - Medicinal chemistry consequences of a TKs analysis Author info Lucia Lintnerová ... [et al.] Author Lintnerová Lucia (11%)
Co-authors Garcia-Caballero Melissa (11%)
Gregáň Fridrich 1944- (11%) UMBFP08 - Katedra chémie
Melicherčík Milan 1948-2015 (11%) UMBFP08 - Katedra chémie
Quesada Ana R. (11%)
Dobiaš Juraj (11%)
Lác Ján (11%)
Sališová Marta (11%)
Boháč Andrej (12%)
Source document European Journal of Medicinal Chemistry. Vol. 72 (2014), pp. 146-159. - Paris : Elsevier Masson SAS, 2014 Keywords medicinálna chémia angiogenéza - angiogenesis kinase inhibitors protein-kinase angiogenesis Language English Country France systematics 53 Public work category ADC No. of Archival Copy 30112 Repercussion category LU, Wen - LI, Pengfei - SHAN, Yuanyuan - SU, Ping - WANG, Jinfeng - SHI, Yaling - ZHANG, Jie. Discovery of biphenyl-based VEGFR-2 inhibitors. Part 3: Design, synthesis and 3D-QSAR studies. In Boorganic & medicinal chemistry. ISSN 0968-0896, 2015, vol. 23, no. 5, pp. 1044-1054.
STAGG, Brian C. - UEHARA, Hironori - LAMBERT, Nathan - RAI, Ruju - GUPTA, Isha S. - RADMALL, Bryce R. - BATES, Taylor - AMBATI, Balamurali Krishna. Morpholino-mediated isoform modulation of vascular endothelial growth factor receptor-2 (VEGFR2) reduces colon cancer xenograft growth. In Cancers. ISSN 2072-6694, 2014, vol. 6, no. 4, pp. 2330-2342.
Catal.org. BB301 - Univerzitná knižnica Univerzity Mateja Bela v Banskej Bystrici Database xpca - PUBLIKAČNÁ ČINNOSŤ References PERIODIKÁ-Súborný záznam periodika Title Návrh štruktúr a syntéza inhibítorov tumorovej neovaskularizácie s VEGFR-2 receptorovou selektivitou Author info Lucia Lintnerová ... [et al.] Author Lintnerová Lucia (40%)
Co-authors Gregáň Fridrich 1944- (10%) UMBFP08 - Katedra chémie
Melicherčík Milan 1948-2015 (10%) UMBFP08 - Katedra chémie
Boháč Andrej (30%)
Sališová Marta (10%)
Source document Študentská vedecká konferencia Prírodovedeckej fakulty UK v Bratislave : zborník recenzovaných príspevkov, Bratislava, 28. apríl 2010. S. 725-729. - Bratislava : Univerzita Komenského, Prírodovedecká fakulta, 2010 / Halgoš Jozef ; Študentská vedecká konferencia Prírodovedeckej fakulty UK vedecká konferencia Keywords inhibítory inhibítory tumorovej neovaskularizácie receptorová selektivita VEGFR2 receptor Language Slovak Country Slovak Republic systematics 544 Public work category AFD No. of Archival Copy 23177 Catal.org. BB301 - Univerzitná knižnica Univerzity Mateja Bela v Banskej Bystrici Database xpca - PUBLIKAČNÁ ČINNOSŤ Title Design and synthesis of sym and asym bispyridine analogues of 1Y6A inhibitor Author info Lucia Lintnerová ... [et al.] Author Lintnerová Lucia (20%)
Co-authors Sališová Marta (16%)
Boháč Andrej (16%)
Gregáň Fridrich 1944- (16%) UMBFP08 - Katedra chémie
Melicherčík Milan 1948-2015 (16%) UMBFP08 - Katedra chémie
Medveď Miroslav 1971- (16%) UMBFP08 - Katedra chémie
Source document COST Action CM0602 : inhibitors of angiogenesis: design, synthesis, and biological exploitation (ANGIOKEM) : 3rd Workshop, Favignana, 16 - 18 October 2009. S. 11. - Milano : University of Milano, 2009 ; COST Action CM06023rd workshop Keywords syntéza - syntézy - synthesis inhibítory dizajn - design inhibitors Language English Country Italy systematics 54 Public work category AFK No. of Archival Copy 23176 Catal.org. BB301 - Univerzitná knižnica Univerzity Mateja Bela v Banskej Bystrici Database xpca - PUBLIKAČNÁ ČINNOSŤ